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Home - Products - Chromatin/Epigenetic - Histone Demethylase - LSD1-IN-7 benzenesulfonate

LSD1-IN-7 benzenesulfonate

CAS No. 2097523-60-7

LSD1-IN-7 benzenesulfonate( CC-90011 benzenesulfonate )

Catalog No. M23947 CAS No. 2097523-60-7

LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 113 In Stock
10MG 178 In Stock
25MG 312 In Stock
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Biological Information

  • Product Name
    LSD1-IN-7 benzenesulfonate
  • Note
    Research use only, not for human use.
  • Brief Description
    LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
  • Description
    LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
  • In Vitro
    ——
  • In Vivo
    Animal Model:BALB/c nude mice bearing small cell lung carcinoma (SCLC)Dosage:5 mg/kg Administration:Oral administration; daily; for 30 days Result:Showed a tumor growth inhibition (TGI) of 78% at 5 mg/kg with nobody weight loss.
  • Synonyms
    CC-90011 benzenesulfonate
  • Pathway
    Chromatin/Epigenetic
  • Target
    Histone Demethylase
  • Recptor
    LSD1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2097523-60-7
  • Formula Weight
    609.64
  • Molecular Formula
    C30H29F2N5O5S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:60mg/ml(98.42mM; Need ultrasonic)
  • SMILES
    N#CC1=CC=C(C(N=C(N2CCC(N)CC2)N3C)=C(C4=CC=C(OC)C(F)=C4)C3=O)C=C1F.O=S(C5=CC=CC=C5)(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Young K. Chen, et al. Compositions comprising an inhibitor of lysine specific demethylase-1. WO2017079670A1.
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